PROTAC BET degrader-2

 CAS No.: 2093388-33-9  Cat No.: BP-400046 4.5  

PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression.

PROTAC BET degrader-2

Structure of 2093388-33-9

Quality
Assurance

Worldwide
Delivery

24/7 Customer
Support
Category
PROTAC
Molecular Formula
C41H42N10O6
Molecular Weight
770.84

* For research and manufacturing use only. Not for human or clinical use.

SizePriceStockQuantity
-- $-- In stock

Looking for different specifications? Click to request a custom quote!

Capabilities & Facilities

  • mg to g scale for early stage;
  • CDMO and CMO support.
  • 24/7 customer service;
  • 100% quality assurance;
  • Efficient global delivery;
  • Over 95% customer satisfaction.
Popular Publications Citing BOC Sciences Products
Solubility
H2O : < 0.1 mg/mL (insoluble); DMSO : 50 mg/mL (64.86 mM; Need ultrasonic)
Storage
Powder<br/>-20°C<br/>3 years<br/><br/><br/> <br/>4°C<br/>2 years<br/><br/><br/>In solvent<br/>-80°C<br/>6 months<br/><br/><br/> <br/>-20°C<br/>1 month
Shipping
Room temperature in continental US; may vary elsewhere
Synonyms
PROTAC BET degrader 2; 4-[(5-cyclopropyl-2-ethylpyrazol-3-yl)amino]-7-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propyl]-6-methoxy-9H-pyrimido[4,5-b]indole-2-carboxamide
InChI Key
LKCUEUQTTCOYPW-UHFFFAOYSA-N
InChI
InChI=1S/C41H42N10O6/c1-5-51-32(18-28(48-51)23-11-12-23)44-37-35-25-17-31(56-4)26(34-20(2)49-57-21(34)3)16-29(25)43-36(35)46-38(47-37)40(54)42-15-7-9-22-8-6-10-24-27(22)19-50(41(24)55)30-13-14-33(52)45-39(30)53/h6,8,10,16-18,23,30H,5,7,9,11-15,19H2,1-4H3,(H,42,54)(H,45,52,53)(H2,43,44,46,47)
Canonical SMILES
CCN1C(=CC(=N1)C2CC2)NC3=NC(=NC4=C3C5=CC(=C(C=C5N4)C6=C(ON=C6C)C)OC)C(=O)NCCCC7=C8CN(C(=O)C8=CC=C7)C9CCC(=O)NC9=O

Stock concentration: *
Desired final volume: *
Desired concentration: *

L

* Our calculator is based on the following equation:
Concentration (start) x Volume (start) = Concentration (final) x Volume (final)
It is commonly abbreviated as: C1V1 = C2V2

Calculate
* Total Molecular Weight:
g/mol
Tip: Chemical formula is case sensitive. C22H30N4O √ c22h30n40 ╳
g/mol
g
Historical Records: FKBP12 PROTAC dTAG-13 | PROTAC Sirt2 Degrader-1 | PROTAC BET degrader-2

Related Product Recommendations

In Stock Purity: 0.98 Hot
Nexturastat A
Nexturastat A

CAS: 1403783-31-2
In Stock Purity: 0.98 Hot
Alisertib
Alisertib

CAS: 1028486-01-2
In Stock Purity: ≥95% Hot
Propargyl-PEG5-acid
Propargyl-PEG5-acid

CAS: 1245823-51-1
In Stock Purity: >98% Hot
DCC-2618
DCC-2618

CAS: 1225278-16-9
In Stock Purity: 95% Hot
Propargyl-PEG2-Tos
Propargyl-PEG2-Tos

CAS: 145916-41-2
In Stock Purity: >95% Hot
Amine-PEG3-Desthiobiotin
Amine-PEG3-Desthiobiotin

CAS: 2237234-71-6
BOC Sciences Support

Please contact us with any specific requirements and we will get back to you as soon as possible.


  • Verification code

We invite you to contact us at or through our contact form above for more information about our services and products.

USA
  • International:
  • US & Canada (Toll free):
  • Email:
  • Fax:
UK
Germany
Copyright © 2025 BOC Sciences. All Rights Reserved.
Inquiry Basket
Loading......
Delete selected Go to checkout