Structure | Catalog | Product Name | CAS | E3 Ligase | Target | Inquiry |
---|---|---|---|---|---|---|
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BPL-202093 | (2S,4R)-1-((S)-2-(tert-Butyl)-14-(4-(((4-((3-chloro-4-fluorophenyl)amino)-6-((E)-4-(piperidin-1-yl)but-2-enamido)quinazolin-7-yl)oxy)methyl)-1H-1,2,3-triazol-1-yl)-4-oxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
EGFR |
Inquiry | |
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BPL-202094 | PROTAC EGFR Degrader 2 | VHL |
EGFR |
Inquiry | |
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BPL-202095 | N1-[4-[(2-Aminophenyl)carbamoyl]phenyl]-N9-[(S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methylthiazol-5-yl)benzyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]nonanediamide | 2669785-72-0 | VHL |
HDAC1 |
Inquiry |
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BPL-202096 | N1-(4-((2-Aminophenyl)carbamoyl)phenyl)-N10-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)decanediamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202097 | N1-(4-((2-Aminophenyl)carbamoyl)phenyl)-N11-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)undecanediamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202098 | N1-(4-((2-Aminophenyl)carbamoyl)phenyl)-N14-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)tetradecanediamide | 2669785-73-1 | VHL |
HDAC1 |
Inquiry |
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BPL-202099 | (2S,4R)-1-((S)-2-(2-((9-((4-((2-Aminophenyl)carbamoyl)phenyl)amino)-9-oxononyl)oxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | 2669785-75-3 | VHL |
HDAC1 |
Inquiry |
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BPL-202100 | JPS014 | 2669785-76-4 | VHL |
HDAC1 |
Inquiry |
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BPL-202101 | (2S,4R)-1-((S)-2-(2-((6-(2-((4-((2-Aminophenyl)carbamoyl)phenyl)amino)-2-oxoethoxy)hexyl)oxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | 2669785-74-2 | VHL |
HDAC1 |
Inquiry |
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BPL-202102 | JPS016 | 2669785-77-5 | VHL |
HDAC1 |
Inquiry |
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BPL-202103 | (2S,4R)-1-((S)-2-(2-(2-(2-((4-((2-Aminophenyl)carbamoyl)phenyl)amino)-2-oxoethoxy)ethoxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202104 | (2S,4R)-1-((S)-14-((4-((2-Aminophenyl)carbamoyl)phenyl)amino)-2-(tert-butyl)-4,14-dioxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202105 | N1-(4-((2-Aminophenyl)carbamoyl)phenyl)-N14-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)-3,6,9,12-tetraoxatetradecanediamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202106 | (2S,4R)-1-((S)-2-(4-(4-(4-((4-((2-Aminophenyl)carbamoyl)phenyl)amino)-4-oxobutyl)piperazin-1-yl)butanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202107 | N1-(4-((2-Amino-4-fluorophenyl)carbamoyl)phenyl)-N9-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)nonanediamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202108 | N1-(4-((2-Amino-4-fluorophenyl)carbamoyl)phenyl)-N12-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)dodecanediamide | 2669785-78-6 | VHL |
HDAC1 |
Inquiry |
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BPL-202109 | (2S,4R)-1-((S)-14-((4-((2-Amino-4-fluorophenyl)carbamoyl)phenyl)amino)-2-(tert-butyl)-4,14-dioxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202110 | (2S,4R)-1-((S)-2-(2-((9-(2-((4-((2-Amino-4-fluorophenyl)carbamoyl)phenyl)amino)-2-oxoethoxy)nonyl)oxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | 2669785-79-7 | VHL |
HDAC1 |
Inquiry |
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BPL-202111 | N1-(4-((2-Amino-5-(thiophen-2-yl)phenyl)carbamoyl)phenyl)-N9-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)nonanediamide | VHL |
HDAC1 |
Inquiry | |
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BPL-202112 | N1-(4-((2-Amino-5-(thiophen-2-yl)phenyl)carbamoyl)phenyl)-N12-((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)dodecanediamide | VHL |
HDAC1 |
Inquiry |