Structure | Catalog | Product Name | CAS | E3 Ligase | Target | Inquiry |
---|---|---|---|---|---|---|
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BPL-201073 | WH174 | VHL |
HDAC6 |
Inquiry | |
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BPL-201074 | WH167 | VHL |
HDAC6 |
Inquiry | |
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BPL-201075 | WH221 | VHL |
HDAC6 |
Inquiry | |
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BPL-201076 | WH212 | VHL |
HDAC6 |
Inquiry | |
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BPL-201077 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(8-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)octyl)acetamide | 2097971-03-2 | CRBN |
BRD9 |
Inquiry |
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BPL-201078 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(1-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-2-oxo-7,10,13-trioxa-3-azahexadecan-16-yl)acetamide | 2097971-06-5 | CRBN |
BRD9 |
Inquiry |
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BPL-201079 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(6-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)hexyl)acetamide | 2097971-07-6 | CRBN |
BRD9 |
Inquiry |
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BPL-201080 | N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)-7-(4-(2-(1'-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetyl)-[4,4'-bipiperidin]-1-yl)-2-oxoethoxy)-3-methoxyphenyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridine-2-carboximidamide | 2097509-52-7 | CRBN |
BRD9 |
Inquiry |
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BPL-201081 | (2S,4R)-1-((S)-2-(tert-Butyl)-17-(4-(2-(N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | 2097971-09-8 | VHL |
BRD9 |
Inquiry |
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BPL-201082 | (2S,4R)-1-((S)-2-(tert-Butyl)-14-(4-(2-(N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-4,13-dioxo-6,9-dioxa-3,12-diazatetradecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | 2097971-15-6 | VHL |
BRD9 |
Inquiry |
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BPL-201083 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)amino)octyl)acetamide | 2097509-23-2 | CRBN |
BRD9 |
Inquiry |
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BPL-201084 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)octyl)acetamide | 2097509-46-9 | CRBN |
BRD9 |
Inquiry |
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BPL-201085 | 2-(4-(2-(N-(1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)octyl)acetamide | 2097509-20-9 | CRBN |
BRD4 |
Inquiry |
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BPL-201086 | 2-((2,6-Dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)benzyl)(methyl)amino)-N-(6-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)amino)hexyl)acetamide | 2170679-40-8 | CRBN |
BRD9 |
Inquiry |
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BPL-201087 | 2-((2,6-Dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)benzyl)(methyl)amino)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)octyl)acetamide | CRBN |
BRD9 |
Inquiry | |
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BPL-201088 | (2S,4R)-1-((S)-18-(tert-Butyl)-1-(2,6-dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)phenyl)-2-methyl-4,16-dioxo-8,11,14-trioxa-2,5,17-triazanonadecan-19-oyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | VHL |
BRD9 |
Inquiry | |
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BPL-201089 | 2-((2,6-Dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)benzyl)(methyl)amino)-N-(8-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)octyl)acetamide | 2170679-44-2 | CRBN |
BRD9 |
Inquiry |
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BPL-201090 | (S)-2-((2S,3R)-3-Amino-2-hydroxy-4-phenylbutanamido)-4-methyl-N-(2-(2-(2-((4-(6-methylbenzo[d]thiazol-2-yl)phenyl)amino)ethoxy)ethoxy)ethyl)pentanamide | 2133321-59-0 | cIAP1 |
Htt |
Inquiry |
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BPL-201091 | (S)-2-((2S,3R)-3-Amino-2-hydroxy-4-phenylbutanamido)-N-(2-(2-(2-((2-((E)-(4-(dimethylamino)phenyl)diazenyl)benzo[d]thiazol-6-yl)oxy)ethoxy)ethoxy)ethyl)-4-methylpentanamide | 2766855-40-5 | cIAP1 |
Htt |
Inquiry |
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BPL-201092 | TMX-1117 | 2488752-67-4 | CRBN |
CDK2 |
Inquiry |